Drug Delivery

Chemical Name:Endomorphin-2-d4Synonyms:L-Tyrosyl-L-prolyl-L-phenylalanyl-L-phenylalaninamide-d4; 12: PN: WO2008052043 SEQID: 11 claimed protein; 1: PN:WO2010004535 PAGE: 30 claimed protein-d4; 2: PN: EP1782819 PAGE-d4: 14 claimed protein; 2: PN: US20110065648 SEQID-d4: 2 claimed protein-d4; 2: PN:WO2011034659 SEQID-d4: 2 claimed protein-d4; 40: PN-d4: WO2005016244 PAGE: 68 claimed protein-d4Alternate CAS #:141801-26-5Molecular Formula:C₃₂H₃₃D₄N₅O₅Molecular Weight:575.69Category:Standards; Isotopic Labeled Analogues; Pharmaceutical/API Drug Impurities/Metabolites;Applications:Isotope labelled Endomorphin-2 is […]

Chemical Name:Enalaprilat Acyl Glucuronide-d5Synonyms:(2S,3S,4S,5R,6S)-6-(((S)-1-((S)-2-(((S)-1-Carboxy-3-phenylpropyl)amino)propanoyl)pyrrolidine-2-carbonyl)oxy)-3,4,5-trihydroxytetrahydro-2H-pyran-2-carboxylic Acid-d5Molecular Formula:C₂₄H₂₇D₅N₂O₁₁Molecular Weight:529.55Category:Standards; Isotopic Labeled Analogues; Pharmaceutical/API Drug Impurities/Metabolites;Applications:Enalaprilat Acyl Glucuronide-d5 is the isotope labelled analog of Enalaprilat Acyl Glucuronide. Enalaprilat Acyl Glucuronide is an acyl glucuronide metabolite of enalapril (E555250). Enalapril is an antihypertensive. An angiotensin-converting enzyme (ACE) inhibitor.References:Tocco, D.J., et al.: Drug Metab. Dispos., 10, 15 (1982), Cohen, M.L., […]

Chemical Name:ent-Emtricitabine Triphosphate Triethylammonium SaltSynonyms:P-[[(2S,4R)-5-(4-Amino-5-fluoro-2-oxo-1(2H)-pyrimidinyl)-1,3-oxathiolan-2-yl]methyl] Ester Triphosphoric Acid Triethylammonium Salt; (2S-cis)-P-[[5-(4-Amino-5-fluoro-2-oxo-1(2H)-pyrimidinyl)-1,3-oxathiolan-2-yl]methyl] Ester Triphosphoric Acid Triethylammonium Salt; Triphosphoric Acid Deriv. 1,3-Oxathiolane Triethylammonium SaltMolecular Formula:C₈H₁₃FN₃O₁₂P₃S . (C₆H₁₅N)ₓMolecular Weight:487.19 . (101.19)xCategory:Standards; Enzyme Activators and Inhibitors;Applications:ent-Emtricitabine Triphosphate Triethylammonium Salt is a metabolite of ent-Emtricitabine (E525005). The free acid, ent-Emtricitabine Triphosphate inhibits the prodn. of full-length minus-strand DNA in an […]

Chemical Name:Emodin 8-O-β-D-(6’-O-Malonylglucoside)Synonyms:8-[[6-O-(2-Carboxyacetyl)-β-D-glucopyranosyl]oxy]-1,6-dihydroxy-3-methyl-9,10-anthracenedioneCAS Number:928262-58-2Molecular Formula:C₂₄H₂₂O₁₃Molecular Weight:518.42Category:Standards; Pharmaceutical/API Drug Impurities/Metabolites;Applications:Emodin 8-O-β-D-(6’-O-malonylglucoside) is a metabolite of emodin (E523000).References:Pan, X., et al.: Biochem. Eng. J., 5, 173 (2000), Srinivas, G., et al.: Eur. J. Pharmacol., 473, 117 (2003), Xiang, H., et al.: Chin. Pharm. J., 40, 96 (2005), Mokhtarani, B., et al.: Biochem. Eng. J., 38, 241 (2008),To […]

Chemical Name:Eliglustat (SR) Diastereomer-D15Synonyms:N-((1R,2S)-1-(2,3-Dihydrobenzo[b][1,4]dioxin-6-yl)-1-hydroxy-3-(pyrrolidin-1-yl)propan-2-yl)octanamide;Alternate CAS #:1092472-65-5Molecular Formula:C₂₃H₂₁D₁₅N₂O₄Molecular Weight:419.64Category:Research Tools; Molecular Biology; Enzyme Activators and Inhibitors; Pharmaceutical/API Drug Impurities/Metabolites;Applications:Eliglustat (SR) Diastereomer-D15 is a labelled isomer of Eliglustat (E508030); a specific and potent inhibitor of glucosylceramide synthase.References:Lukina Elena., et al.: Blood, 116, 893 (2010); McEachern Kerry Anne., et al.: Mol Genet Metab Rep., 91, 259 (2007);To ensure the stability of our […]

Chemical Name:Eliglustat (SR) DiastereomerSynonyms:N-[(1S,2R)-2-(2,3-Dihydro-1,4-benzodioxin-6-yl)-2-hydroxy-1-(1-pyrrolidinylmethyl)ethyl]octanamide;CAS Number:1092472-65-5Molecular Formula:C₂₃H₃₆N₂O₄Molecular Weight:404.54Category:Research Tools; Molecular Biology; Enzyme Activators and Inhibitors; Pharmaceutical/API Drug Impurities/Metabolites;Applications:Eliglustat Rs-​Isomer is an isomer of Eliglustat (E508030); a specific and potent inhibitor of glucosylceramide synthase.References:Lukina Elena., et al.: Blood, 116, 893 (2010); McEachern Kerry Anne., et al.: Mol Genet Metab Rep., 91, 259 (2007);To ensure the stability of our products, the efficient […]

Chemical Name:(4S)-EdoxabanSynonyms:N1-(3,5-Dichloropyridin-2-yl)-N2-((1S,2R,4S)-4-(dimethylcarbamoyl)-2-(5-methyl-4,5,6,7-tetrahydrothiazolo[5,4-c]pyridine-2-carboxamido)cyclohexyl)oxalamide; Edoxaban Impurity 42Molecular Formula:C₂₄H₂₉Cl₂N₇O₄SMolecular Weight:582.5Applications:(4S)-Edoxaban is an impurity of Edoxaban (E555520). Edoxaban is an anticoagulant drug which acts as a direct factor Xa inhibitor.References:Ruff, C., et al.: Am. Heart J., 160, 635 (2010); Ogata, K., et al.: J. Clin. Pharm., 50, 73 (2010);To ensure the stability of our products, the efficient express delivery […]

Chemical Name:(5R)-tert-Butyl EdoxabanSynonyms:tert-Butyl ((1S,2R,5R)-2-(2-((5-chloropyridin-2-yl)amino)-2-oxoacetamido)-5-(dimethylcarbamoyl)cyclohexyl)carbamateCAS Number:1255529-33-9Molecular Formula:C₂₁H₃₀ClN₅O₅Molecular Weight:467.95Applications:(5R)-tert-Buty Edoxaban is an impurity of Edoxaban (E555520). Edoxaban is an anticoagulant drug which acts as a direct factor Xa inhibitor.References:Ruff, C., et al.: Am. Heart J., 160, 635 (2010); Ogata, K., et al.: J. Clin. Pharm., 50, 73 (2010);To ensure the stability of our products, the efficient express […]

Chemical Name:(1R, 5S)-tert-Butyl EdoxabanSynonyms:tert-Butyl ((1R,2R,5S)-2-(2-((5-chloropyridin-2-yl)amino)-2-oxoacetamido)-5-(dimethylcarbamoyl)cyclohexyl)carbamateCAS Number:480451-98-7Molecular Formula:C₂₁H₃₀ClN₅O₅Molecular Weight:467.95Applications:(1R, 5S)-tert-Buty Edoxaban is an impurity of Edoxaban (E555520). Edoxaben is an anticoagulant drug which acts as a direct factor Xa inhibitor.References:Ruff, C., et al.: Am. Heart J., 160, 635 (2010); Ogata, K., et al.: J. Clin. Pharm., 50, 73 (2010);To ensure the stability of our products, the […]

Chemical Name:Efonidipine Hydrochloride MonoethanolateSynonyms:5-(5,5-Dimethyl-2-oxido-1,3,2-dioxaphosphorinan-2-yl)-1,4-dihydro-2,6-dimethyl-4-(3-nitrophenyl)-3-pyridinecarboxylic Acid 2-[Phenyl(phenylmethyl)amino]ethyl Ester Hydrochloride Monoethanolate; 3-Pyridinecarboxylic Acid, 5-(5,5-Dimethyl-1,3,2-dioxaphosphorinan-2-yl)-1,4-dihydro-2,6-dimethyl-4-(3-nitrophenyl)-, 2-[Phenyl(phenylmethyl)amino]ethyl Ester, P-Oxide, Monohydrochloride, compd. with Ethanol (1:1); 5-(5,5-Dimethyl-2-oxido-1,3,2-dioxaphosphorinan-2-yl)-1,4-dihydro-2,6-dimethyl-4-(3-nitrophenyl)-3-pyridinecarboxylic Acid, 2-[Phenyl(phenylmethyl)amino]ethylEster, Monohydrochloride, compd. withEhanol (1:1) (9CI); 1,3,2-Dioxaphosphorinane, 3-Pyridinecarboxylic Acid deriv.; Ethanol, compd. with 2-[Phenyl(phenylmethyl)amino]ethyl 5-(5,5-dimethyl-1,3,2-dioxaphosphorinan-2-yl)-1,4-dihydroCAS Number:111011-76-8Molecular Formula:C₃₄H₃₈N₃O₇P • C ₂H₆O • HClMolecular Weight:631.66 + 46.07 + 36.46Category:Standards; Enzyme Activators and Inhibitors;Applications:Efonidipine Hydrochloride Monoethanolate […]