Drug Delivery

Catalogue Number:B196500Chemical Name:1-Benzhydryl-3-cyanoazetidineSynonyms:1-(Diphenylmethyl)-3-azetidinecarbonitrile; 3-Cyano-1-(diphenylmethyl)azetidine;CAS Number:36476-86-5Molecular Formula:C₁₇H₁₆N₂Appearance:White SolidMelting Point:153-155°CMolecular Weight:248.34Storage:-20°CSolubility:Chloroform (Slightly), Methanol (Slightly)Category:Research Tools; Enzyme Activators and Inhibitors;Applications:A proline analog and proline formation inhibitor.References:Sheers, M., et al.: Int. J. Parasitology, 12, 47 (1982),To ensure the stability of our products, the efficient express delivery service will be used. We also guarantee that the products will be shipped […]

Catalogue Number:B195500Chemical Name:1-Benzhydrylazetidin-3-olSynonyms:1-(Diphenylmethyl)-3-hydroxyazetinide; 1-(Diphenylmethyl)-3-azetidinol; 1-(Diphenylmethyl)-3-azetidinol; NSC 319045;CAS Number:18621-17-5Molecular Formula:C₁₆H₁₇NOAppearance:Off-White to Pale Yellow SolidMelting Point:107-110°CMolecular Weight:239.32Storage:-20°CSolubility:Chloroform (Slightly), Methanol (Slightly)Category:Research Tools; Enzyme Activators and Inhibitors;Applications:It is used to identify inhibitors of CYP 3A4.References:Kulkarni., et al.: Pestic. Biochem. Physiol., 6, 183 (1976),To ensure the stability of our products, the efficient express delivery service will be used. We also […]

Catalogue Number:B195305Chemical Name:3-Bromo-2,5,6-trifluoroanilineSynonyms:3-Bromo-2,5,6-trifluorobenzenamine;CAS Number:1269440-68-7Molecular Formula:C₆H₃BrF₃NMolecular Weight:226Category:Building Blocks; Miscellaneous;Applications:3-Bromo-2,5,6-trifluoroaniline is a useful research chemical for organic synthesis and other chemical processes.References:Huang, S., et al.: From PCT Int. Appl. (2011), WO 2011025927 A1 20110303To ensure the stability of our products, the efficient express delivery service will be used. We also guarantee that the products will be shipped […]

Catalogue Number:B195000Chemical Name:Benzhydryl BromideSynonyms:1,1′-(Bromomethylene)bisbenzene; Bromomethylene)dibenzene; 1,1′-(Bromomethylene)bis[benzene]; 1-[Bromo(phenyl)methyl]benzene; Bromodiphenylmethane; Diphenylbromomethane; Diphenylmethyl Bromide; NSC 39226; α-Bromodiphenylmethane; α-Phenylbenzyl BromideCAS Number:776-74-9Molecular Formula:C₁₃H₁₁BrAppearance:Pale Brown to Brown Low-Melting SolidMelting Point:>36°C (dec.)Molecular Weight:247.13Storage:4°CSolubility:Chloroform, Methanol (Slightly)Category:Building Blocks; Miscellaneous;Applications:Benzhydryl Bromide is used as a reagent in the synthesis of O-(triazolyl)methyl carbamates as a novel and potent class of fatty acid amide hydrolase (FAAH) inhibitors.Not […]

Catalogue Number:B194875Chemical Name:1-Benzhydrylazetidine-3-carboxylic AcidSynonyms:1-(Diphenylmethyl)azetidine-3-carboxylic Acid;CAS Number:36476-87-6Molecular Formula:C₁₇H₁₇NO₂Appearance:Brown Crystalline SolidMelting Point:182-190°CMolecular Weight:267.32Solubility:DMF, DMSOCategory:Building Blocks; Amino Acids;Applications:A useful intermediate in the synthesis of polypeptides.To ensure the stability of our products, the efficient express delivery service will be used. We also guarantee that the products will be shipped in the box with layers of tapes to protect them […]

Catalogue Number:B194843Chemical Name:1-Benzo[b]thien-4-yl-piperazineSynonyms:1-Benzo[b]thiophen-4-ylpiperazine; 4-(1-Piperazinyl)benzo[b]thiopheneCAS Number:846038-18-4Molecular Formula:C₁₂H₁₄N₂SAppearance:Pale Brown SolidMelting Point:>75ºC (dec.)Molecular Weight:218.32Storage:-20°CSolubility:DMSO (Slightly), Methanol (Slightly)Category:Building Blocks; Miscellaneous;Applications:is an intermediate in synthesizing Brexpiprazole 5-1H-Quinolin-2-one (B677428), an impurity of Brexpiprazole (B677385), which is a drug candidate useful in treatment and prevention of mental disorders including CNS disorders.References:Yamashita, H., et al.: PCT Int. Appl., WO 2006112464 A1 20061026 (2006)To ensure the stability of […]

Catalogue Number:B194842Chemical Name:3-(Benzo[d]thiazol-2-yl)-7-(diethylamino)-2H-chromene-2-thioneSynonyms:3-(2-Benzothiazolyl)-7-(diethylamino)-2H-1-benzopyran-2-thione;CAS Number:211228-18-1Molecular Formula:C₂₀H₁₈N₂OS₂Molecular Weight:366.5Category:Research Tools; Materials; Dyes;Applications:3-(Benzo[d]thiazol-2-yl)-7-(diethylamino)-2H-chromene-2-thione is used in the making of coumarin and anthraquinone dyes with large absorption coefficient and little fluorescence for guest-host type liquid crystal displays.References:Iwanaga, H., et al.: Bull. Chem. Soc. Jpn, 71, 1719 (1998); Iwanaga, H., et al.: From Jpn. Kokai Tokkyo Koho (1998), JP 10316970 A 19981202To ensure the stability of […]

Catalogue Number:B194840Chemical Name:1-Benzo[b]thien-4-yl-piperazine MonohydrochlorideCAS Number:913614-18-3Alternate CAS #846038-18-4 free amineMolecular Formula:C₁₂H₁₅ClN₂SAppearance:White SolidMelting Point:>250°C (dec.)Molecular Weight:254.78Storage:4°CSolubility:DMSO (Slightly, Heated), Methanol (Very Slightly)Category:Building Blocks;Applications:1-Benzo[b]thien-4-yl-piperazine is the starting material to prepare piperazine-substituted benzothiophenes useful in treatment and prevention of mental disorders including CNS disorders.References:Yamashita, H., et al.: PCT Int. Appl., WO 2006112464 A1 20061026 (2006)To ensure the stability of our products, the efficient express […]

Catalogue Number:B194270Chemical Name:Benzyl (2R)-2-Chlorocarbonylpyrrolidine-1-carboxylateSynonyms:(R)-2-(Chlorocarbonyl)-1-pyrrolidinecarboxylic Acid Phenylmethyl Ester; N-(Benzyloxycarbonyl)-D-proline Chloride; N-Cbz-D-proline Chloride;CAS Number:61350-62-7Molecular Formula:C₁₃H₁₄ClNO₃Molecular Weight:267.71Category:Standards; Pharmaceutical/API Drug Impurities/Metabolites;Applications:Benzyl (2R)-2-Chlorocarbonylpyrrolidine-1-carboxylate is an intermediate used in the synthesis of 5-Ethyl-3-[[(2R)-1-methyl-2-pyrrolidinyl]methyl]-1H-indole (E924900), which is an impurity of Eletriptan (E505000), a serotonin 5-HTIB/ID receptor agonist and an anti-migraine agent.References:Madasu, S. B., et al.: Beilstein. J. Org. Chem., 8, 1400 (2012); […]

Catalogue Number:B194260Chemical Name:1-Benzyl-2-chloro-1H-indole-3-carboxaldehydeSynonyms:1-Benzyl-2-chloroindole-3-carbaldehyde; 2-Chloro-1-(phenylmethyl)-1H-indole-3-carboxaldehydeCAS Number:77655-46-0Molecular Formula:C₁₆H₁₂ClNOAppearance:Yellow SolidMolecular Weight:269.73Storage:-20°CSolubility:Chloroform, DichloromethaneCategory:Standards; Miscellaneous;Applications:1-Benzyl-2-chloro-1H-indole-3-carboxaldehyde is an intermediate in synthesizing 2,3,4,10-Tetrahydro-1H-indolo[2,3-b][1,8]naphthyridin-2-ol (T294270), a derivative of 6,7,8,9-Tetrahydro-7-hydroxy-5-methyl-3-phenyl-pyrido[3’,2’:4,5]imidazo[1,2-a]pyrimidinium Chloride (H957770), a carcinogen used in the study of intestinal bacteria metabolism. Created through the heat processing of food.References:Vanhaecke, L.. et al.: Food Chem. Toxicol., 46, 140 (2008)To ensure the stability of our products, […]