Drug Delivery

Catalogue Number:B197845Chemical Name:5-[2-[4-(1,2-Benzisothiazol-3-yl)-1-piperazinyl]ethyl]-6-chloro-1,3-dihydro-3-(1-methylethylidene)-2H-indol-2-oneCAS Number:684269-12-3Molecular Formula:C₂₄H₂₅ClN₄OSMolecular Weight:453Category:Standards; Pharmaceutical/API Drug Impurities/Metabolites;Applications:5-[2-[4-(1,2-Benzisothiazol-3-yl)-1-piperazinyl]-1-hydroxyethyl]-6-chloro-1,3-dihydro-2H-indol-2-one is an impurity of Ziprasidone (Z48500), which is a combined serotonin (5HT2) and dopamine (D2) receptor antagonist. Used as an antipsychotic.References:Bench, C.J., et al.: Psychopharmacology, 112, 308 (1993), Goldstein, J.M.: Exp. Opin. Invest. Drugs, 4, 291 (1995)To ensure the stability of our products, the efficient express […]

Catalogue Number:B197840Chemical Name:7-(1H-Benzimidazol-2-yl)-6-(phenylamino)thieno[3,2-d]pyrimidin-4(3H)-oneSynonyms:7-(1H-Benzimidazol-2-yl)-6-(phenylamino)thieno[3,2-d]pyrimidin-4(1H)-oneCAS Number:496971-05-2Molecular Formula:C₁₉H₁₃N₅OSMolecular Weight:359.4Category:Standards; Pharmaceutical/API Drug Impurities/Metabolites;Applications:7-(1H-Benzimidazol-2-yl)-6-(phenylamino)thieno[3,2-d]pyrimidin-4(3H)-one is a derivative of thieno[3,2-d]pyrimidin-4(3H)-one, a compound used in the identification of novel PARP-1 inhibitors by structure-based virtual screening.References:Hannigan, K., et al.: Bioorg. Med. Chem. Lett., 23, 5790 (2013)To ensure the stability of our products, the efficient express delivery service will be used. We also guarantee […]

Catalogue Number:B197825Chemical Name:1H-Benzimidazole-4-methyl-2-propyl-6-carboxylic AcidSynonyms:4-Methyl-2-propyl-6-benzimidazolecarboxylic Acid; 7-Methyl-2-propyl-1H-benzimidazole-5-carboxylic Acid; Telmisartan Benzimidazole Acid Impurity:Impurity:Telmisartan Benzimidazole Acid Impurity:CAS Number:152628-03-0Molecular Formula:C₁₂H₁₄N₂O₂Appearance:Pale Yellow to Tan PowderMelting Point:>286ºC (dec.)Molecular Weight:218.25Storage:-20°CSolubility:DMSO, MethanolCategory:Building Blocks; Miscellaneous;Applications:1H-Benzimidazole-4-methyl-2-propyl-6-carboxylic Acid (cas# 152628-03-0) is a compound useful in organic synthesis.To ensure the stability of our products, the efficient express delivery service will be used. We also guarantee that the […]

Catalogue Number:B197817Chemical Name:5-Bromopyridin-2(1H)-one-3,4,6-d3Synonyms:5-​Bromopyridin-​3,​4,​6-​d3-​2-​olCAS Number:2241872-50-2Molecular Formula:C₅HBrD₃NOMolecular Weight:177.02Category:Building Blocks; Isotopic Labeled Analogues;Applications:5-Bromopyridin-2(1H)-one-3,4,6-d3 is a useful isotopic research intermediate.To ensure the stability of our products, the efficient express delivery service will be used. We also guarantee that the products will be shipped in the box with layers of tapes to protect them against damage. The extremely low temperature […]

Catalogue Number:B197655Chemical Name:BMS-919373Synonyms:5-[5-phenyl-4-[[(pyridin-2-yl)methyl]amino]quinazolin-2-yl]pyridine-3-sulfonamide;CAS Number:1272353-82-8Molecular Formula:C₂₅H₂₀N₆O₂SMolecular Weight:468.53Category:Research Tools; Standards; Molecular Biology; Enzyme Activators and Inhibitors; Pharmaceutical/API Drug Impurities/Metabolites;Applications:BMS-919373 (CAS# 1272353-82-8) is an intermediate in the synthesis of clinical candidate 5-(5-phenyl-4-(pyridin-2-ylmethylamino)quinazolin-2-yl)pyridine-3-sulfonamide as a selective IKur inhibitor for potential treatment of atrial fibrillation.References:Gunaga, P., et al.: J. Med. Chem., 60, 3795 (2017)To ensure the stability of our products, […]

Catalogue Number:B197050Chemical Name:4-(1H-Benzimidazol-2-yl)-3-(2,4-dihydroxyphenyl)-1H-pyrazole-5-propanoic AcidCAS Number:1217314-90-3Molecular Formula:C₁₉H₁₆N₄O₄Molecular Weight:364.35Category:Research Tools;Applications:4-(1H-Benzimidazol-2-yl)-3-(2,4-dihydroxyphenyl)-1H-pyrazole-5-propanoic Acid is novel inhibitor of DNA gyrase B with low micromolar antigyrase activity.References:Brvar, M., et al.: Bioorg. Med. Chem., 20, 958 (2010);To ensure the stability of our products, the efficient express delivery service will be used. We also guarantee that the products will be shipped in the […]

Catalogue Number:B197040Chemical Name:Benzimidazole 2-Sulfonic AcidSynonyms:2-Benzimidazolesulfonic Acid; 1H-Benzimidazole-2-sulfonic Acid; Rabeprazole Sulfonic Acid Impurity:Impurity:Rabeprazole Sulfonic Acid Impurity:CAS Number:40828-54-4Molecular Formula:C₇H₆N₂O₃SAppearance:Off-White to Pale Beige SolidMelting Point:>230°C (dec.)Molecular Weight:198.2Storage:4°CCategory:Building Blocks; Miscellaneous;Applications:Benzimidazole 2-Sulfonic Acid is a versatile reactant used in the preparation of bis(benzimidazol-2-yl)amines with antitrichinellosis activity.References:Mavrova, A., et al.: Bioorg. Med. Chem., 15, 6291 (2007);To ensure the stability of our […]

Catalogue Number:B197021Chemical Name:Benzimidazole-4,5,6,7-d4CAS Number:64531-29-9Alternate CAS #51-17-2Molecular Formula:C₇H₂D₄N₂Molecular Weight:122.16Category:Building Blocks; Isotopic Labeled Analogues; Miscellaneous;Applications:Benzimidazole-4,5,6,7-d4 (CAS# 64531-29-9) is a useful isotopically labeled research compound.To ensure the stability of our products, the efficient express delivery service will be used. We also guarantee that the products will be shipped in the box with layers of tapes to protect them […]

Catalogue Number:B197020Chemical Name:1H-Benzimidazole-5-carboxylic AcidSynonyms:1H-Benzimidazole-6-carboxylic Acid; 5-Benzimidazolecarboxylic Acid; 3H-Benzimidazole-5-carboxylic Acid; 3H-Benzo[d]imidazole-5-carboxylic Acid; 5-Carboxybenzimidazole; Benzimidazole-6-carboxylic Acid;CAS Number:15788-16-6Molecular Formula:C₈H₆N₂O₂Appearance:Off-White to Pale Yellow SolidMelting Point:>300°C (dec.)Molecular Weight:162.15Storage:4°CSolubility:DMSO (Slightly), Methanol (Slightly, Heated)Category:Building Blocks; Miscellaneous;Applications:A benzimidazole derivative that exhibits corrosion inhibiting properties against strong acids.References:Popova, A., Bull. Electrochem., 23, 137 (2007), Popova, A., et al.: Corros. Sci., 46, 1333 (2004),To ensure […]

Catalogue Number:B197010Chemical Name:BenzilideSynonyms:3,3,6,6-Tetraphenyl-1,4-dioxane-2,5-dione; NSC 403081; NSC 677243CAS Number:467-32-3Molecular Formula:C₂₈H₂₀O₄Appearance:White to Off-White SolidMelting Point:194-196°CMolecular Weight:420.46Storage:4°CSolubility:Chloroform (Slightly), Ethyl Acetate (Slightly)Category:Building Blocks; Pharmaceutical/API Drug Impurities/Metabolites;Applications:Benzilide is an impurity of Trospium (T892800), a tropine derivative with anticholinergic activity and is used to treat urinary incontinence.References:Antweiler, H., et al.: Arzneim.-Forsch., 16, 1581 (1966), Lux, G., et al.: Fortschr. Med., 96, […]