Drug Delivery

Catalogue Number:B198200Chemical Name:Benzoctamine HydrochlorideSynonyms:N-Methyl-9,10-ethanoanthracene-9(10H)-methanamine Hydrochloride; 9-(Methylaminomethyl)-9,10-dihydro-9,10-ethanoanthracene Hydrochloride; Ba-30803; Tacitin; Tracitin;CAS Number:10085-81-1Alternate CAS #17243-39-9Molecular Formula:C₁₈H₂₀ClNAppearance:White to Off-White SolidMelting Point:>271°C (dec.)Molecular Weight:285.81Storage:4°C, HygroscopicSolubility:DMSO (Slightly), Methanol (Slightly)StabilityHygroscopicCategory:Standards; Pharmaceutical/API Drug Impurities/Metabolites;Applications:Anxiolytic.References:Geisler, L., et al.: Arzneim.-Forsch., 20, 957 (1970), Goldenthal, E.I., et al.: Toxicol. Appl. Pharmacol., 18, 185 (1971),To ensure the stability of our products, the efficient express delivery service […]

Catalogue Number:B197952Chemical Name:Benzocaine-d4Synonyms:4-Aminobenzoic Acid-d4 Ethyl Ester; p-Aminobenzoic-d4 Acid Ethyl Ester; Ethyl 4-Aminobenzoate-d4; (p-(Ethoxycarbonyl)(phenyl-d4)mine; 4-(Ethoxycarbonyl)aniline-d4; 4-(Ethoxycarbonyl)(phenyl-d4)amine; 4-Aminobenzoic Acid-d4 Ethyl Ester; 4-Carbethoxyaniline-d4; Aethoform-d4; Amben-d4 Ethyl Ester; Americaine-d4; Anaesthan-syngala-d4;CAS Number:342611-08-9Alternate CAS #unlabelled: 94-09-7Molecular Formula:C₉H₇D₄NO₂Appearance:Off-White to Light Yellow SolidMelting Point:85-870CMolecular Weight:169.21Storage:-20°CSolubility:Chloroform (Slightly), Methanol (Slightly)Category:Standards; Isotopic Labeled Analogues; Pharmaceutical/API Drug Impurities/Metabolites;Applications:Labelled Benzocaine (B202970). Benzocaine is used as an anesthetic (local).References:Ali, […]

Catalogue Number:B197940Chemical Name:Benz[a]anthracene-7,12-dioneSynonyms:1,2-Benzanthraquinone; Benzanthraquinone; 1,2-Benzo-9,10-anthraquinone; Benz[a]anthra-7,12-quinone; Benz[a]anthracene-7,12-quinone; Benzanthracene-7,12-dione; Benzo[a]anthrancene-7,12-dione; C.I. 59000; NSC 7961; Sirius Yellow GCAS Number:2498-66-0Molecular Formula:C₁₈H₁₀O₂Appearance:Light Yellow to Yellow SolidMelting Point:168 – 169°CMolecular Weight:258.27Storage:4°CSolubility:Chloroform (Slightly), Methanol (Slightly)Category:Standards; Pharmaceutical/API Drug Impurities/Metabolites;Applications:Benz[a]anthracene-7,12-dione is a polycyclic aromatic hydrocarbon that is present in the emission soot of biomass fuels combustion. Benz[a]anthracene-7,12-dione is an urban air contaminant and […]

Catalogue Number:B197930Chemical Name:2-​[[(1R,​2R)​-​2-​[[4-​(1,​2-​Benzisothiazol-​3-​yl)​-​1-​piperazinyl]​methyl]​cyclohexyl]​methyl]​-1H-​isoindole-​1,​3(2H)​-​dioneSynonyms:2-(((1R,2R)-2-((4-(Benzo[d]isothiazol-3-yl)piperazin-1-yl)methyl)cyclohexyl)methyl)isoindoline-1,3-dioneCAS Number:1260025-92-0Molecular Formula:C₂₇H₃₀N₄O₂SAppearance:Yellow SolidMolecular Weight:474.62Solubility:Chloroform, Dichloromethane, Ethyl AcetateCategory:Standards; Pharmaceutical/API Drug Impurities/Metabolites;Applications:2-​[[(1R,​2R)​-​2-​[[4-​(1,​2-​Benzisothiazol-​3-​yl)​-​1-​piperazinyl]​methyl]​cyclohexyl]​methyl]​-1H-​isoindole-​1,​3(2H)​-​dione is an intermediate in synthesizing Lurasidone Opened Imide (L474935), an impurity in the synthesis of Lurasidone (L474920) which is antipsychotic used for treatment of schizophrenia.References:Ishiyama, T., et al.: Eur. J. Pharmacol., 572, 160 (2007); Cole, P., et al.: Drugs of the Fut., […]

Catalogue Number:B197925Chemical Name:BenznidazoleSynonyms:2-Nitro-N-(phenylmethyl)-1H-imidazole-1-acetamide; N-Benzyl-2-nitro-Imidazole-1-acetamide; Benznidazole; Benzonidazol; Benzonidazole; N-Benzyl-2-nitroimidazol-1-yl-acetamide; NSC 299972; Radanil; Ro 07-1051; Ro 71051; Rochagan;CAS Number:22994-85-0Molecular Formula:C₁₂H₁₂N₄O₃Appearance:White to Off-White SolidMelting Point:188-190°CMolecular Weight:260.25Storage:4°CSolubility:DMSO (Slightly), Methanol (Slightly)Category:Standards; Pharmaceutical/API Drug Impurities/Metabolites;Applications:Benznidazole (BNZ) is traditionally used to treat Chagas disease caused by Trypanosoma cruzi. The drugs used for the treatment of this disease, Nifurtimox and Benznidazole, are toxic […]

Catalogue Number:B197905Chemical Name:4-(1,2-Benzisothiazol-3-yl)-1-piperazinecarboxylic Acid 1,1-Dimethylethyl EsterCAS Number:131779-46-9Molecular Formula:C₁₆H₂₁N₃O₂SAppearance:Yellow SolidMolecular Weight:319.42Solubility:DCMCategory:Building Blocks; Miscellaneous;Applications:4-(1,2-Benzisothiazol-3-yl)-1-piperazinecarboxylic Acid 1,1-Dimethylethyl Ester is an intermediate in the synthesis of Ziprasidone (Z485010) related compounds.References:Huang, M., et al.: Clin. Pharmacol. Ther., 54, 257 (1993),To ensure the stability of our products, the efficient express delivery service will be used. We also guarantee that the products […]

Catalogue Number:B197900Chemical Name:1,2-Benzisoxazole-5-carboxylic AcidSynonyms:Benzo[d]isoxazole-5-carboxylic AcidCAS Number:933744-95-7Molecular Formula:C₈H₅NO₃Molecular Weight:163.13Category:Building Blocks; Miscellaneous;Applications:1,2-Benzisoxazole-5-carboxylic Acid is used as a reagent in the synthesis of pyrazolopyrimidinone compounds for the inhibition of PAS Kinase (PASK) activity.References:Mccall, J., et al.: PCT Int. Appl. WO 2014066795 A1 20140501. May 1, 2014To ensure the stability of our products, the efficient express delivery service will be used. We also […]

Catalogue Number:B197875Chemical Name:3-(1,2-Benzisothiazolyl) Ziprasidone (Ziprasidone Impurity E)Synonyms:3-(1,2-Benzisothiazol-3-yl)-5-[2-[4-(1,2-benzisothiazol-3yl)-1-piperazinyl]ethyl]-6-chloro-1,3-dihydro-2H-indol-2-one; Ziprasidone EP Impurity E;Impurity:Ziprasidone EP Impurity ECAS Number:1159977-04-4Molecular Formula:C₂₈H₂₄ClN₅OS₂Molecular Weight:546.11Category:Standards; Pharmaceutical/API Drug Impurities/Metabolites;Applications:3-(1,2-Benzisothiazolyl) Ziprasidone is an impurity of Ziprasidone. Ziprasidone is a combined serotonin (5HT2) and dopamine (D2) receptor antagonist. Used as an antipsychotic.References:Bench, C.J., et al.: Psychopharmacology, 112, 308 (1993), Goldstein, J.M.: Exp. Opin. Invest. Drugs, 4, […]

Catalogue Number:B197865Chemical Name:(3aR,7aR)-4′-(1,2-Benzisothiazol-3-yl)octahydro-spiro[2H-isoindole-2,1′-piperazinium] MethanesulfonateSynonyms:Spiro[2H-isoindole-2,1′-piperazinium], (3aR,7aR)-4′-(1,2-benzisothiazol-3-yl)octahydro-spiro[2H-isoindole-2,1′-piperazinium] Monomethanesulfonate; (3aR-trans)-4′-(1,2-benzisothiazol-3-yl)octahydro-spiro[2H-isoindole-2,1′-piperazinium] Monomethanesulfonate; Lurasidone Impurity B;CAS Number:186204-37-5Molecular Formula:C19H26N3S•CH3O2SOAppearance:White to Off-White SolidMelting Point:224 – 228°CMolecular Weight:423.58Storage:-20°CSolubility:Chloroform (Slightly), Methanol (Slightly)Category:Standards; Pharmaceutical/API Drug Impurities/Metabolites;Applications:(3aR,7aR)-4′-(1,2-Benzisothiazol-3-yl)octahydro-spiro[2H-isoindole-2,1′-piperazinium] Methanesulfonate (B197865) is a useful synthetic intermediate for Lurasidone Hydrochloride (L474920), an antipsychotic used for treatment of schizophrenia.References:Zhang, P., et al.: Huagong Shikan, 27, 5 (2013)To ensure the stability […]

Catalogue Number:B197860Chemical Name:BenziodaroneSynonyms:(2-Ethyl-3-benzofuranyl)(4-hydroxy-3,5-diiodophenyl)methanone; Algocor; Cardivix; 2-Ethyl-3-(3,5-diiodo-4-hydroxybenzoyl)-3-coumarone; L 2329; NSC 82133; 2-Ethyl-3-(3,5-diiodo-4-hydroxybenzoyl)benzofuran; 2329 Labaz; Amplivix; Corofam; Dilafurane; Retrangor; 2-Ethyl-3-(4-hydroxy-3,5-diiodobenzoyl)benzofuran; Coronal-Crinos; Dila-Vasal; 2-Ethyl-3-(4-hydroxy-3,5-diiodobenzoyl)coumarone;CAS Number:68-90-6Molecular Formula:C₁₇H₁₂I₂O₃Appearance:Pale Beige to Beige SolidMelting Point:160-164°C (dec.)Molecular Weight:518.08Storage:4°CSolubility:Chloroform (Slightly), DMSO (Slightly), Ethyl Acetate (Slightly)Category:Standards; Pharmaceutical/API Drug Impurities/Metabolites;Applications:A uricosuric drug. It is used to effectively to control hyperuricemia in renal transplantation.References:Lemieux, G. et al.: […]