Chemical Name:6’-Hydroxy N-Desisopropyl Delavirdine-d8Synonyms:N-[2-[[4-(3-Amino-1,6-dihydro-6-oxo-2-pyridinyl)-1-piperazinyl]carbonyl]-1H-indol-5-yl]methanesulfonamide-d8; 1-(3-Amino-1,6-dihydro-6-oxo-2-pyridinyl)-4-[[5-[(methylsulfonyl)amino]-1H-indol-2-yl]carbonyl]piperazine-d8Alternate CAS #:Unlabelled: 188780-41-8Molecular Formula:C₁₉H₁₄D₈N₆O₄SMolecular Weight:438.53Category:Standards; Isotopic Labeled Analogues; Pharmaceutical/API Drug Impurities/Metabolites;Applications:6’-Hydroxy N-Desisopropyl Delavirdine-d8 is the isotope labelled analog of 6’-Hydroxy N-Desisopropyl Delavirdine (H936540); a metabolite of Delavirdine (D230625) which is a bisheteroarylpiperazine (BHAP) reverse transcriptase inhibitor.References:Dueweke, T.J., et al.: Antimicrob. Ag. Chemother., 37, 1127 (1993); Althaus, I.W., et al.: Biochem. […]

Chemical Name:p-Hydroxyatazanavir-d4Synonyms:3,12-Bis(1,1-dimethylethyl)-8-hydroxy-4,11-dioxo-9-(p-hydroxyphenyl-d4-methyl)-6-[[4-(2-pyridinyl)phenyl]methyl]-dimethyl EsterAlternate CAS #:Unlabelled CAS# N/AMolecular Formula:C₃₈H₄₈D₄N₆O₈Molecular Weight:724.88Category:Building Blocks; Isotopic Labeled Analogues;Applications:p-Hydroxyatazanavir-d4 is the labeled analog of p-Hydroxyatazanavir (H828175), a metabolite of Atazanavir (A790051), a novel azapeptide HIV protease inhibitor (PI). Antiviral.References:Palella, F.J. Jr., et al.: N. Engl. J. Med., 338(13), 853 (1998); Nolan, D., et al.: Drugs, 63(23), 2555 (2003); Musial, B.L., et […]

Chemical Name:5-Hydroxyfraxetin 8-beta-D-GlucosideSynonyms:5,7-Dihydroxy-6-methoxy-8-(((2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)tetrahydro-2H-pyran-2-yl)oxy)-2H-chromen-2-one; 5,7-Dihydroxy-6-methoxycoumarin 8-β-D-Glucoside; 5,7-Dihydroxy-6-methoxycoumarin 8-β-D-GlucopyranosideMolecular Formula:C₁₆H₁₈O₁₁Molecular Weight:386.31Category:Standards; Pharmaceutical/API Drug Impurities/Metabolites; Carbohydrates and Oligosaccharides;Applications:5-Hydroxyfraxetin 8-β-D-Glucoside is a derivative of Fraxetin (F763960); a coumarin compound with anti-oxidant and anti-inflammatory activity. It also acts as a protective agent against hyperuricemia and renal dysfunction.References:Witaicenis, A. et al.: Phytomed. 21, 240 (2014); Chen, X. et al.: Int. Immunopharm., […]

Chemical Name:4-Hydroxy Atorvastatin Acyl-β-D-glucuronide 80%, contains up to 20% lactoneSynonyms:(βR,δR)-2-(4-Fluorophenyl)-β,δ-dihydroxy-4-[[(4-hydroxyphenyl)amino]carbonyl]-5-(1-methylethyl)-3-phenyl-1H-pyrrole-1-heptanoic Acid β-D-Glucopyranuronic Acid;Molecular Formula:C₃₉H₄₃FN₂O₁₂Molecular Weight:750.76Category:Standards; Pharmaceutical/API Drug Impurities/Metabolites;Applications:A metabolite of Atorvastatin (A791750).To ensure the stability of our products, the efficient express delivery service will be used. We also guarantee that the products will be shipped in the box with layers of tapes to protect them […]

Chemical Name:Hydroxy Famciclovir-d4Alternate CAS #:unlabelled: 172645-79-3Molecular Formula:C₁₄H₁₅D₄N₅O₅Molecular Weight:341.36Category:Standards; Isotopic Labeled Analogues;Applications:Hydroxy Famciclovir-d4 is the labelled analogue of Hydroxy Famciclovir, which is a Famciclovir (F101125) derivative and may be a useful hepadnaviridae-active antiviral agent.References:Marcuccio, S. M., et al.: PCT Int. Appl. WO 9522330 A1 19950824 (1995)To ensure the stability of our products, the efficient express delivery service will be used. We also guarantee that […]

Chemical Name:4-Hydroxycarbazeran-d4Synonyms:1-(3,4-Dihydro-6,7-dimethoxy-4-oxo-1-phthalazinyl)-4-piperidinyl Ester Ethylcarbamic Acid-d4;Alternate CAS #:Unlabelled: 96724-43-5Molecular Formula:C₁₈H₂₀D₄N₄O₅Molecular Weight:380.43Category:Building Blocks; Isotopic Labeled Analogues;Applications:4-Hydroxycarbazeran-d4 is the isotope labelled analog of 4-Hydroxycarbazeran, a metabolite of Carbazeran (C175790). Carbazeran is known as a phosphodiesterase inhibitor drug that exhibits chronictropic and inotropic effects.References:Kaye, B., et al.: Xenobiotica., 15, 237 (1985); Shahid, M., et al.: Br. J. Pharmacol., 98, 291 […]

Chemical Name:7β-HydroxygliclazideSynonyms:rel-(3aα,5α,6aα)-N-[[(Hexahydro-5-hydroxycyclopenta[c]pyrrol-2(1H)-yl)amino]carbonyl]-4-methyl-benzenesulfonamide; 5-Hydroxy-hexahydro-cyclopenta[c]pyrrole BenzenesulfonamideCAS Number:96860-48-9Molecular Formula:C₁₅H₂₁N₃O₄SMolecular Weight:339.41Category:Standards; Pharmaceutical/API Drug Impurities/Metabolites;Applications:7β-Hydroxygliclazide is a metabolite of Gliclazide (G409875) which is a a sulfonylurea hypoglycemic agent used as an antidiabetic.References:Duhault, J., et al.: Arzneimittel-Forsch., 22, 1686 (1972), Holmes, B., et al.: Drugs, 27, 301 (1984),To ensure the stability of our products, the efficient express delivery service will be […]

Chemical Name:13-Hydroxy CabotegravirSynonyms:(3S,11aR)-N-(2,4-Difluorobenzyl)-2,6-dihydroxy-3-methyl-5,7-dioxo-2,3,5,7,11,11a-hexahydrooxazolo[3,2-a]pyrido[1,2-d]pyrazine-8-carboxamideMolecular Formula:C₁₉H₁₇F₂N₃O₆Molecular Weight:421.35Category:Standards; Enzyme Activators and Inhibitors; Pharmaceutical/API Drug Impurities/Metabolites;Applications:13-Hydroxy Cabotegravir is a metabolite of Cabotegravir (C050100). Cabotegravir is a long acting HIV-1 integrase inhibitor with action against a broad range of HIV subtypes.References:Yoshinaga, T. et al.: Antimicrob, Agents Chemother., 59, 397 (2015); Andrews, C. et al.: Sci. Transl. Med., 7, 270 (2015)To […]

Chemical Name:13-Hydroxy Cabotegravir-d3Synonyms:(3S,11aR)-N-(2,4-Difluorobenzyl)-2,6-dihydroxy-3-methyl-5,7-dioxo-2,3,5,7,11,11a-hexahydrooxazolo[3,2-a]pyrido[1,2-d]pyrazine-8-carboxamide-d3Molecular Formula:C₁₉H₁₄D₃F₂N₃O₆Molecular Weight:424.37Category:Standards; Isotopic Labeled Analogues; Enzyme Activators and Inhibitors; Pharmaceutical/API Drug Impurities/Metabolites;Applications:13-Hydroxy Cabotegravir-d3 is the labelled form of 13-Hydroxy Cabotegravir. 13-Hydroxy Cabotegravir is a metabolite of Cabotegravir (C050100). Cabotegravir is a long acting HIV-1 integrase inhibitor with action against a broad range of HIV subtypes.References:Yoshinaga, T. et al.: Antimicrob, Agents Chemother., 59, […]

Chemical Name:24-Hydroxy CabotegravirSynonyms:(3S,11aR)-N-(2,4-Difluoro-3-hydroxybenzyl)-6-hydroxy-3-methyl-5,7-dioxo-2,3,5,7,11,11a-hexahydrooxazolo[3,2-a]pyrido[1,2-d]pyrazine-8-carboxamideMolecular Formula:C₁₉H₁₇F₂N₃O₆Molecular Weight:421.35Category:Standards; Enzyme Activators and Inhibitors; Pharmaceutical/API Drug Impurities/Metabolites;Applications:24-Hydroxy Cabotegravir is a metabolite of Cabotegravir (C050100). Cabotegravir is a long acting HIV-1 integrase inhibitor with action against a broad range of HIV subtypes.References:Yoshinaga, T. et al.: Antimicrob, Agents Chemother., 59, 397 (2015); Andrews, C. et al.: Sci. Transl. Med., 7, 270 (2015)To […]