Chemical Name:(R)-5-BromocoerulescineSynonyms:(3R)-5-bromo-1′-methylspiro[3H-indole-3,3′-pyrrolidin]-2(1H)-one;Molecular Formula:C₁₂H₁₃BrN₂OMolecular Weight:281.15Category:Standards; Pharmaceutical/API Drug Impurities/Metabolites;Applications:(R)-5-Bromocoerulescine, is a derivative of Coerulescine, which is an oxindole that can be found in the plant Horsfieldia superba, and it has analgesic effects.References:Jossang, A. et al.: J. Org. Chem. 56 (23): 6527–6530; Lakshmaiah, G. et al.: J. Org. Chem.64 (5): 1699–1704;To ensure the stability of our products, the […]

Chemical Name:(3R, 4R)-1-Boc-4-methylpiperidin-3-ol-d3Molecular Formula:C₁₁H₁₈D₃NO₃Molecular Weight:218.31Category:Standards; Isotopic Labeled Analogues;Applications:(3R, 4R)-1-Boc-4-methylpiperidin-3-ol-d3 is an isotope labelled analog of (3R, 4R)-1-Boc-4-methylpiperidin-3-ol (B667885).To ensure the stability of our products, the efficient express delivery service will be used. We also guarantee that the products will be shipped in the box with layers of tapes to protect them against damage. The extremely […]

Chemical Name:(3S,5R)-1-tert-Butyl 3-Methyl 5-(((Benzyloxy)carbonyl)amino)piperidine-1,3-dicarboxylateSynonyms:(3S,5R)-5-[[(Phenylmethoxy)carbonyl]amino]-1,3-piperidinedicarboxylic Acid 1-(1,1-Dimethylethyl) 3-Methyl EsterCAS Number:1448902-04-2Molecular Formula:C₂₀H₂₈N₂O₆Molecular Weight:392.45Category:Building Blocks;Applications:(3S,5R)-1-tert-Butyl 3-Methyl 5-(((Benzyloxy)carbonyl)amino)piperidine-1,3-dicarboxylate is used in the preparation of (3S,5R)-5-(2,2-dimethyl-5-oxo-4-phenylpiperazin-1-yl)piperidine-3-carboxamides as orally active renin inhibitors.References:Mori, Y., et. al.: Bioorg. Med. Chem., 21, 5907 (2013)To ensure the stability of our products, the efficient express delivery service will be used. We also guarantee that the products […]

Chemical Name:BP-1-108Synonyms:4-​[[(4-​Cyclohexylphenyl)​methyl]​[2-​[methyl[(2,​4,​6-​trimethylphenyl)​sulfonyl]​amino]​acetyl]​amino]​-​2-​hydroxy-Benzoic AcidCAS Number:1334492-85-1Molecular Formula:C₃₂H₃₈N₂O₆SMolecular Weight:578.72Category:Standards; Pharmaceutical/API Drug Impurities/Metabolites;Applications:BP-1-108 is a small molecule STAT5-SH2 domain inhibitor used in antileukemia treatment.References:Page, B. et al.: J. Med. Chem., 53, 1047 (2012); Page, B. et al.: Bioorg. Med. Chem. Lett., 21, 5605 (2011);To ensure the stability of our products, the efficient express delivery service will be used. We […]

Chemical Name:tert-Butyl ((3R,4S)-4-phenethylpyrrolidin-3-yl)carbamateCAS Number:1260602-53-6Molecular Formula:C₁₇H₂₆N₂O₂Molecular Weight:290.4Category:Building Blocks;Applications:tert-Butyl ((3R,4S)-4-phenethylpyrrolidin-3-yl)carbamate, is used in the synthesis of pharmaceutical and biologically active compounds. It can be used in the synthesis of Pteridine reductase (PTR1) inhibitors, using for the treatment of African Sleeping Sickness and the Leishmaniases.References:Tulloch, L.B. et al.: J. Med. Chem., 53, 221 (2010);To ensure the stability of […]

Chemical Name:Brilacidin TetrahydrochlorideSynonyms:PMX 30063 Tetrahydrochloride; N4,N6-Bis[3-[[5-[(aminoiminomethyl)amino]-1-oxopentyl]amino]-2-[(3R)-3-pyrrolidinyloxy]-5-(trifluoromethyl)phenyl]-4,6-pyrimidinedicarboxamide HydrochlorideCAS Number:1224095-99-1Molecular Formula:C₄₀H₅₄Cl₄F₆N₁₄O₆Molecular Weight:1082.75Category:Standards; Pharmaceutical/API Drug Impurities/Metabolites;Applications:Brilacidin Tetrahydrochloride is a defensin mimetic.References:Scott, R.W.: Am. Biotech. Lab., 27, 16 (2009)To ensure the stability of our products, the efficient express delivery service will be used. We also guarantee that the products will be shipped in the box with layers of tapes […]

Chemical Name:(S)-tert-Butyl 1-((2S,3S)-3-Amino-4-(tert-butoxy)-2-((tert-butyldimethylsilyl)oxy)-4-oxobutyl)azetidine-2-carboxylateMolecular Formula:C₂₂H₄₄N₂O₅SiMolecular Weight:444.68Category:Building Blocks; Chiral Molecules; Amino Acids; Miscellaneous;Applications:(S)-tert-Butyl 1-((2S,3S)-3-Amino-4-(tert-butoxy)-2-((tert-butyldimethylsilyl)oxy)-4-oxobutyl)azetidine-2-carboxylate is an intermediate for the synthesis of Mugineic Acid Ammonium Salt (M792005). Mugineic Acid, a possible phytosiderophore of graminaceous plants, has iron chelation potency and antioxidant activity.References:Takagi, S., et al.: J. Plant. Nutr., 7, 469 (1984); Das, P., et al.: Nat. Prod. Res., […]

Chemical Name:B498358Synonyms:2-Methyl-4,5-oxazoledicarboxylic Acid; 2-Methyloxazole-4,5-dicarboxylic AcidCAS Number:855404-45-4Molecular Formula:C₆H₅NO₅Molecular Weight:171.11Category:Building Blocks; Miscellaneous;Applications:2-Methyl-1,3-oxazole-4,5-dicarboxylic Acid can be useful in the study of oxazole synthesis from ethyl acetoacetate.References:Cornforth, J. W., et al.: J. Chem. Soc., 93 (1953)To ensure the stability of our products, the efficient express delivery service will be used. We also guarantee that the products will be shipped […]

Chemical Name:Bisphenol A Monosulfate Disodium-13C12Synonyms:Sodium 4-(2-(4-Oxidophenyl-1,2,3,4,5,6-13C6)propan-2-yl)phenyl-1,2,3,4,5,6-13C6 SulfateMolecular Formula:C₃¹³C₁₂H₁₄Na₂O₅SMolecular Weight:364.23Category:Standards; Isotopic Labeled Analogues; Pharmaceutical/API Drug Impurities/Metabolites;Applications:Labelled Bisphenol A Monosulfate Disodium is a derivative of Bisphenol A (B519495), a monomer used for policarbonate and epoxy resins; exhibits estrogenic activity. BPA is also used as a building block in polycarbonate bottles and in the epoxy-resin liners of metal […]

Chemical Name:1,8-Bis(4-((1,4,8,11-tetraazacyclotetradecan-1-yl)methyl)benzyl)-1,4,8,11-tetraazacyclotetradecaneSynonyms:Plexifor Impurity II;CAS Number:414858-02-9Molecular Formula:C₄₆H₈₄N₁₂Molecular Weight:805.24Category:Standards; Enzyme Activators and Inhibitors; Pharmaceutical/API Drug Impurities/Metabolites;Applications:1,8-Bis(4-((1,4,8,11-tetraazacyclotetradecan-1-yl)methyl)benzyl)-1,4,8,11-tetraazacyclotetradecane is an impurity of Plerixafor (P580500), a hematopoietic stem cell (HSC) mobilizer that inhibits the CXCR4 chemokine receptor and blocks binding of its ligand, stromal cell-derived factor-1-α (SDF-1-α). This agent was approved on Dec. 15, 2008, as treatment in combination with […]