Chemical Name:3-Chlorobalipramine-d6 MaleateSynonyms:3-Chloro-5-[3-(dimethylamino)propyl]-5H-dibenz[b,f]azepine-d6 ; 3-Chloro-N,N-dimethyl-5H-Dibenz[b,f]azepine-5-propanamine-d6Alternate CAS #:Unlabelled: 2095-42-3Molecular Formula:C₂₃H₁₉D₆ClN₂O₄Molecular Weight:434.95Category:Standards; Isotopic Labeled Analogues; Pharmaceutical/API Drug Impurities/Metabolites;Applications:Isotope labelled 3-Chlorobalipramine is an halogenated metabolite of Balipramine (B115700), a tricyclic anti-depressant and an impurity of imipramine (I465980).References:Bickel, M.H., et al.: Int. J. Neuropharmacol., 3, 611 (1964); Craig, P.N., et al.: J. Org. Chem., 26, 135 (1961);To ensure the […]

Chemical Name:Chloro Efavirenz(Mixture of Diastereomers)Synonyms:(4S)-6-Chloro-4-[(2-chlorocyclopropyl)ethynyl]-1,4-dihydro-4-(trifluoromethyl)-2H-3,1-benzoxazin-2-one;CAS Number:1322625-98-8Molecular Formula:C₁₄H₈Cl₂F₃NO₂Molecular Weight:350.12Category:Standards; Pharmaceutical/API Drug Impurities/Metabolites;Applications:Efavirenz (E425000) derivative.To ensure the stability of our products, the efficient express delivery service will be used. We also guarantee that the products will be shipped in the box with layers of tapes to protect them against damage. The extremely low temperature products will be […]

Chemical Name:1-Chloroethyl (2-(6-Methoxy-3-(1-pyridin-2-yl)ethyl)-1H-inden-2-yl)ethyl)(methyl)carbamateMolecular Formula:C₂₃H₂₇ClN₂O₃Molecular Weight:414.93Category:Standards; Pharmaceutical/API Drug Impurities/Metabolites;Applications:1-Chloroethyl (2-(6-Methoxy-3-(1-pyridin-2-yl)ethyl)-1H-inden-2-yl)ethyl)(methyl)carbamate is an intermediate used in the synthesis of 6-Hydroxy-N-demethyldimethidene (H934110), which is a metabolite of the antihistaminic drug dimethindene.References:Rudolf, J., Blaschke, G.: Enantiomer, 4, 317 (1999)To ensure the stability of our products, the efficient express delivery service will be used. We also guarantee that the products […]

Chemical Name:N-[3-Chloro-4-[(3-fluorophenyl)methoxy]phenyl]-6-[5-[[2-((1-Oxyl-2,2,5,5-tetramethylpyrroline-3-yl)carbamido)ethyl]amino]methyl]-2-furanyl]-4-quinazolinamineSynonyms:Demethylsulfonyl Lapatinib 1-Oxyl-2,2,5,5-tetramethyl-Æ3-pyrroline deriv;Molecular Formula:C₃₇H₃₇ClFN₆O₄Molecular Weight:684.18Category:Standards; Enzyme Activators and Inhibitors; Pharmaceutical/API Drug Impurities/Metabolites;Applications:N-[3-Chloro-4-[(3-fluorophenyl)methoxy]phenyl]-6-[5-[[2-((1-Oxyl-2,2,5,5-tetramethylpyrroline-3-yl)carbamido)ethyl]amino]methyl]-2-furanyl]-4-quinazolinamine is an analog of Lapatinib Ditosylate (L175800) which acts as a reversible dual inhibitor of ErbB1 and ErbB2 tyrosine kinases. Antineoplastic.References:Kim, T.E., et al.: Drugs, 6, 886 (2003), Wood, E.R., et al.: Cancer Res., 64, 6652 (2004), Spector, N.L., et al.: […]

Chemical Name:7α-Chloro-16α-methyl PrednisoloneSynonyms:(7α,11β,16α)-7-Chloro-11,17,21-trihydroxy-16-methylpregna-1,4-diene-3,20-dione; 7α-Chloro-16α-methylprednisolone; Alclometasone; Alclomethasone;CAS Number:67452-97-5Molecular Formula:C₂₂H₂₉ClO₅Molecular Weight:408.92Category:Standards; Pharmaceutical/API Drug Impurities/Metabolites; Steroids;Applications:A metabolite of Alclometasone dipropionate (A514580); a synthetic glucocorticoid steroid for topical use in dermatology as anti-inflammatory, antipruritic, antiallergic, antiproliferative and vasoconstrictive agent.References:Aoyama, S. et al.: Drug Metab. Disp., 18, 409 (1990); Green, M.J. et al.: J. Steroid Biochem., 11, 61 (1979); De, […]

Chemical Name:Cefcanel Daloxate HydrochlorideSynonyms:[6R-[6α,7β(R*)]]-L-Alanine 2-[[2-[[(5-methyl-2-oxo-1,3-dioxol-4-yl)methoxy]carbonyl]-3-[[(5-methyl-1,3,4-thiadiazol-2-yl)thio]methyl]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-en-7-yl]amino]-2-oxo-1-phenylethyl Ester Monohydrochloride; KY 109; 1R)-2-[[(6R,7R)-2-[[(5-Methyl-2-oxo-1,3-dioxol-4-yl)methoxy]carbonyl]-3-[[(5-methyl-1,3,4-thiadiazol-2-yl)thio]methyl]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-en-7-yl]amino]-2-oxo-1-phenylethyl Ester L-Alanine MonohydrochlorideCAS Number:92602-21-6Alternate CAS #:free base: CAS 97275-40-6Molecular Formula:C₂₇H₂₇N₅O₉S₃ •HClMolecular Weight:661.73+(36.46)Category:Standards; Pharmaceutical/API Drug Impurities/Metabolites;Applications:Cefcanel Daloxate Hydrochloride can be used in analytical study for cefcanel determination in human blood plasma and urine by HPLC after administration of, as prodrug.References:Lanbeck-Vallen, K., & Carlqvist, J.: J. Chromatogr-biomed., […]

Chemical Name:Cefepime-D3,13C SulfateSynonyms:1-[[(6R,7R)-7-[[(2Z)-(2-Amino-4-thiazolyl)(methoxyimino)acetyl]amino]-2-carboxy-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-en-3-yl]methyl]-1-methylpyrrolidinium-D3,13C Sulfate (1:1); [6R-[6α,7β(Z)]]-1-[[7-[[(2-Amino-4-thiazolyl)(methoxyimino)acetyl]amino]-2-carboxy-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-en-3-yl]methyl]-1-methylpyrrolidinium-D3,13C Sulfate (1:1)Alternate CAS #:Unlabelled: 107648-78-2/Free Base: 88376-58-3Molecular Formula:C₁₈¹³CH₂₄D₃N₆O₉S₃Molecular Weight:583.66Category:Building Blocks; Isotopic Labeled Analogues;Applications:Cefepime-D3,13C sulfate is a labelled analogue of Cefepine sulfate, a cephalosporin that has antibacterial effects against Gram-positive and Gram-negative bacteria. Cefepime sulfate is used to treat mild to severe bacterial infections.References:Neu, H.: Am. J. Med., 100, 68S […]

Chemical Name:∆2-(E)-Cefpodoxime ProxetilMolecular Formula:C₂₁H₂₇N₅O₉S₂Molecular Weight:557.6Category:Standards; Pharmaceutical/API Drug Impurities/Metabolites;Applications:∆2-(E)-Cefpodoxime Proxetil is derived from (E)-Cefpodoxime Proxetil (C243855), which is the (E)-isomer of Cefpodoxime Proxetil (C243860); an antibacterial and broad spectrum, orally absorbed third generation cephalosporin. The (E)-isomer tends to have less antibacterial activity than the (Z)-isomer.References:Fujimoto, K., et al.: J. Antibiot., 40, 370 (1987); Utsui, Y., et […]

Chemical Name:3-(6-Chloropyrimidin-4-yl)-5-(1-methylcyclopropoxy)-2-((2-(trimethylsilyl)ethoxy)methyl)-2H-indazoleCAS Number:1627093-41-7Molecular Formula:C₂₁H₂₇ClN₄O₂SiMolecular Weight:431Category:Building Blocks; Miscellaneous;Applications:3-(6-Chloropyrimidin-4-yl)-5-(1-methylcyclopropoxy)-2-((2-(trimethylsilyl)ethoxy)methyl)-2H-indazole is a useful intermediate in the development of MLi-​2 (3-​(4-​Pyrimidinyl) Indazole), a potent orally available brain penetrant inhibitor of LRRK2.References:Scott, J. D., et al.: J. Med. Chem., 60, 2983 (2017);To ensure the stability of our products, the efficient express delivery service will be used. We also guarantee that […]

Chemical Name:CandoxatrilSynonyms:cis-4-[[[1-[(2S)-3-[(2,3-Dihydro-1H-inden-5-yl)oxy]-2-[(2-methoxyethoxy)methyl]-3-oxopropyl]cyclopentyl]carbonyl]amino]cyclohexanecarboxylic Acid; UK 79300;CAS Number:123122-55-4Molecular Formula:C₂₉H₄₁NO₇Molecular Weight:515.64Category:Research Tools;Applications:Neutral endopeptidase inhibitor. Used in treatment of congestive heart failure.References:Motwani, J.G., et al.: Clin. Pharmacol. Ther., 54, 661 (1993), Kimmelstiel, C.D., et al.: Cardiology, 87, 46 (1996),To ensure the stability of our products, the efficient express delivery service will be used. We also guarantee that the products […]